http://www.cnr.it/ontology/cnr/individuo/rivista/ID263491
Bioorganic & medicinal chemistry letters
- Label
- Bioorganic & medicinal chemistry letters (literal)
- Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#rivistaDi
- Synthesis of a potential photoactivatable anandamide analog (Articolo in rivista) (Prodotto della ricerca)
- New metabolically stable fatty acid amide ligands of cannabinoid receptors: synthesis and receptor affinity studies (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and enzymatic evaluation of novel partially fluorinated thiol dual ACE/NEP inhibitors (Articolo in rivista) (Prodotto della ricerca)
- Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The homovanillyl moiety (Articolo in rivista) (Prodotto della ricerca)
- Efficient and chemoselective N-acylation of 10-amino-7-ethyl camptothecin with poly(ethylene glycol) (Articolo in rivista) (Prodotto della ricerca)
- Anchimeric assistance effect on regloselective hydrolysis of branched PEGs: a mechanistic investigation (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of All-trans Isomer of Arachidonic Acid and Its Effect on Rabbit Plateled Aggregation (Articolo in rivista) (Prodotto della ricerca)
- Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- 3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- SYNTHESIS OF CARBAPENEMS VIA METALLOIMINES-ESTER ENOLATES CONDENSATION - A NEW SYNTHESIS OF (+)-1-BETA-METHYL PS-5 (Articolo in rivista) (Prodotto della ricerca)
- A novel super-potent neurokinin a receptor antagonist containing dehydroalanine (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Towards novel S-DABOC inhibitors: Synthesis, biological investigation, and molecular modeling studies. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Indolyl-pyrrolone as a new scaffold for Pim1 inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Evidences for complex formation between l-dabPNA and aegPNA (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthetic approaches to DNMT inhibitor SGI-1027 and effects on the U937 leukemia cell line. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- New tetrazole-based selective anandamide uptake inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Kinetic and anion inhibition studies of a beta-carbonic anhydrase (FbiCA 1) from the C-4 plant Flaveria bidentis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and biological evaluation of new potential inhibitors of N-acylethanolamine hydrolyzing acid amidase. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Discovery of novel benzimidazolones as potent non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains. (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological investigation of S-aryl-S-DABO derivatives as HIV-1 inhibitors. (Articolo in rivista) (Prodotto della ricerca)
- Enzymatic regio- and diastereoselective hydrolysis of peracetylated glycerol- and erhythritol-beta-glucosides (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Praziquantel derivatives I: Modification of the aromatic ring. (Articolo in rivista) (Prodotto della ricerca)
- Impurity analysis of retinoic acid samples (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Metabolically labile cannabinoid esters: A 'soft drug' approach for the development of cannabinoid-based therapeutic drugs (Articolo in rivista) (Prodotto della ricerca)
- Tetrahydro-beta-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels. . (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies. (Articolo in rivista) (Prodotto della ricerca)
- Glycosynthase-catalysed syntheses at pH below neutrality. (Articolo in rivista) (Prodotto della ricerca)
- Bradykinin antagonists modified with dipeptide mimetic beta-turn inducers (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase VII is S-glutathionylated without loss of catalytic activity and affinity for sulfonamide inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Effect of acyclic monoterpene alcohols and their derivatives on TRP channels (Articolo in rivista) (Prodotto della ricerca)
- Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: towards the next generation HIV-1 inhibitors (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and evaluation of diverse thio avarol analogs as potential UVB photoprotective candidates (Articolo in rivista) (Prodotto della ricerca)
- Natural and synthetic G-quadruplex interactive berberine derivatives. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and binding affinity at alpha4beta2 and alpha7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- A New Lipophilic Fluorescent Probe for Interaction Studies of Bioactive Lipopeptides with Membrane Models (Articolo in rivista) (Prodotto della ricerca)
- A novel thermophilic glycosynthase that effects branching glycosylation. (Articolo in rivista) (Prodotto della ricerca)
- N-Hydroxyurea as zinc binding group in matrix metalloproteinase inhibition: mode of binding in a complex with MMP-8. (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutants. (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties (Articolo in rivista) (Prodotto della ricerca)
- Novel imidazole-based combretastatin A-4 analogues: Evaluation of their in vitro antitumor activity and molecular modeling study of their binding to the colchicine site of tubulin (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Inhibition of the R1 fragment of the cadmium-containing zeta-class carbonic anhydrase from the diatom Thalassiosira weissflogii with anions. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of Thr200 and Gln92 for obtaining tight-binding inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candidaalbicans and Candida glabrata (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II \"selective\" inhibitor celecoxib. (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of sulfonamides with effective inhibitory action against Porphyromonas gingivalis gamma-carbonic anhydrase (Articolo in rivista) (Prodotto della ricerca)
- Anion inhibition studies of two new beta-carbonic anhydrases from the bacterial pathogen Legionella pneumophila (Articolo in rivista) (Prodotto della ricerca)
- New highly hydrosoluble and not self-aggregated perylene derivatives with three and four polar side chains as G-quadruplex telomere targeting agents and telomerase inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum-The eta-carbonic anhydrases (Articolo in rivista) (Prodotto della ricerca)
- Evidences for complex formation between L-dabPNA and aegPNA (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. (Articolo in rivista) (Prodotto della ricerca)
- Design of novel alpha7-subtype-preferring nicotinic acetylcholine receptor agonists: application of docking and MM-PBSA computational approaches, synthetic and pharmacological studies (Articolo in rivista) (Prodotto della ricerca)
- Investigations of the esterase, phosphatase, and sulfatase activities of the cytosolic mammalian carbonic anhydrase isoforms I, II, and XIII with 4-nitrophenyl esters as substrates (Articolo in rivista) (Prodotto della ricerca)
- CARBONIC ANHYDRASE INHIBITORS: X-RAY CRYSTALLOGRAPHIC STUDIES FOR THE BINDING OF 5-AMINO-1,3,4-THIADIZOLE-2-SULFONAMIDE AND 5-(4-AMINO-3-CHLORO-5-FLUOROPHENYLSULFONAMIDO)-1,3,4-THIADIAZOLE-2-SULFONAMIDE TO HUMAN ISOFORM II (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase inhibitors: Inhibition of human, bacterial, and archaeal isozymes with benzene-1,3-disulfonamides - Solution and crystallographic studies (Articolo in rivista) (Prodotto della ricerca)
- A new cytotoxic tambjamine alkaloid from the Azorean nudibranch Tambja ceutae. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Rational design, synthesis and characterization of potent, drug-like monomeric Smac mimetics as pro-apoptotic anticancer agents (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB(1) receptors. (Articolo in rivista) (Prodotto della ricerca)
- Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB1 receptors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- N-(thiazol-2-yl)-2-thiophene carboxamide derivatives as Abl inhibitors identified by a pharmacophore-based database screening of commercially available compounds. (Articolo in rivista) (Prodotto della ricerca)
- Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents. (Articolo in rivista) (Prodotto della ricerca)
- Soluble polyphenols: synthesis and bioavailability of 3,4',5-tri(alpha-D-glucose-3-O-succinyl)resveratrol. (Articolo in rivista) (Prodotto della ricerca)
- Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes. (Articolo in rivista) (Prodotto della ricerca)
- Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds (Articolo in rivista) (Prodotto della ricerca)
- (-)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels (Articolo in rivista) (Prodotto della ricerca)
- An improved procedure for the synthesis of branched polyethylene glycols (pegs) with the reporter dipeptide Met-bala for protein conjugation (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and anticonvulsant activity of new N-1',N-3'-disubstituted-2'H,3H,5'H-spiro-(2-benzofuran-1,4'-imidazolidine)-2',3,5'-triones (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enantioselective synthesis and vanilloid activity evaluation of 1-â-(p-methoxycinnamoyl)polygodial, an antinociceptive compound from Drymis winteri barks (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- New 1,8-naphthyridine and quinoline derivatives as CB(2) selective agonists (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of new Praziquantel analogues: Potential candidates for the treatment of schistosomiasis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and biological evaluation of novel amides of dopamine with polyunsaturated fatty acids (Articolo in rivista) (Prodotto della ricerca)
- omega-Alkoxy analogues of SAHA(vorinostat) as inhibitors of HDAC: a study of chain-lenght and stereochemical dependence. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Perylene diimides with different side chains are selective in inducing different G-Quadruplex DNA structures and in inhibiting telomerase (Articolo in rivista) (Prodotto della ricerca)
- Anion inhibition study of the beta-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Sulfonamide inhibition studies of the delta-carbonic anhydrase from the diatom Thalassiosira weissflogii (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Sulfonamide inhibition studies of the gamma-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enantioselective synthesis and vanilloid activity evaluation of 1-beta-(p-methoxycinnamoyl)polygodial, an antinociceptive compound from Drymis winteri barks. (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Development of mitochondrial-targeted derivatives o resveratrol. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and alpha4beta2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Discovery of potent nucleotide-mimicking competitive inhibitors of hepatitis C virus NS3 helicase. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enzymatic syntheses and selective hydrolysis of O-b-D-galactopyranosides using a marine mollusc b-galactosidase (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- 5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Selective interactions of perylenederivatives having different side chains with inter- and intramolecular G-quadruplex DNA structures. A correlation with telomerase inhibition (Articolo in rivista) (Prodotto della ricerca)
- Alternative label
- Bioorg. med. chem. lett. (literal)
- Bioorganic and medicinal chemistry letters (literal)
- Bioorganic & medicinal chemistry letters. (literal)
- Language
- Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#issn
- Preferred label
- Bioorganic & medicinal chemistry letters (literal)
- Publisher
- Pergamon, Oxford : GBR (literal)
Incoming links:
- Rivista
- Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies. (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II (Articolo in rivista) (Prodotto della ricerca)
- Evidences for complex formation between l-dabPNA and aegPNA (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Perylene diimides with different side chains are selective in inducing different G-Quadruplex DNA structures and in inhibiting telomerase (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological evaluation of novel amides of dopamine with polyunsaturated fatty acids (Articolo in rivista) (Prodotto della ricerca)
- Efficient and chemoselective N-acylation of 10-amino-7-ethyl camptothecin with poly(ethylene glycol) (Articolo in rivista) (Prodotto della ricerca)
- Anchimeric assistance effect on regloselective hydrolysis of branched PEGs: a mechanistic investigation (Articolo in rivista) (Prodotto della ricerca)
- Enzymatic syntheses and selective hydrolysis of O-b-D-galactopyranosides using a marine mollusc b-galactosidase (Articolo in rivista) (Prodotto della ricerca)
- New metabolically stable fatty acid amide ligands of cannabinoid receptors: synthesis and receptor affinity studies (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of a potential photoactivatable anandamide analog (Articolo in rivista) (Prodotto della ricerca)
- Selective interactions of perylenederivatives having different side chains with inter- and intramolecular G-quadruplex DNA structures. A correlation with telomerase inhibition (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and anticonvulsant activity of new N-1',N-3'-disubstituted-2'H,3H,5'H-spiro-(2-benzofuran-1,4'-imidazolidine)-2',3,5'-triones (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- omega-Alkoxy analogues of SAHA(vorinostat) as inhibitors of HDAC: a study of chain-lenght and stereochemical dependence. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enantioselective synthesis and vanilloid activity evaluation of 1-â-(p-methoxycinnamoyl)polygodial, an antinociceptive compound from Drymis winteri barks (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- New 1,8-naphthyridine and quinoline derivatives as CB(2) selective agonists (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- A new cytotoxic tambjamine alkaloid from the Azorean nudibranch Tambja ceutae. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents. (Articolo in rivista) (Prodotto della ricerca)
- N-(thiazol-2-yl)-2-thiophene carboxamide derivatives as Abl inhibitors identified by a pharmacophore-based database screening of commercially available compounds. (Articolo in rivista) (Prodotto della ricerca)
- Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- A novel thermophilic glycosynthase that effects branching glycosylation. (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors: Inhibition of human, bacterial, and archaeal isozymes with benzene-1,3-disulfonamides - Solution and crystallographic studies (Articolo in rivista) (Prodotto della ricerca)
- Investigations of the esterase, phosphatase, and sulfatase activities of the cytosolic mammalian carbonic anhydrase isoforms I, II, and XIII with 4-nitrophenyl esters as substrates (Articolo in rivista) (Prodotto della ricerca)
- Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Inhibition of the R1 fragment of the cadmium-containing zeta-class carbonic anhydrase from the diatom Thalassiosira weissflogii with anions. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. (Articolo in rivista) (Prodotto della ricerca)
- An improved procedure for the synthesis of branched polyethylene glycols (pegs) with the reporter dipeptide Met-bala for protein conjugation (Articolo in rivista) (Prodotto della ricerca)
- Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB1 receptors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and evaluation of diverse thio avarol analogs as potential UVB photoprotective candidates (Articolo in rivista) (Prodotto della ricerca)
- A New Lipophilic Fluorescent Probe for Interaction Studies of Bioactive Lipopeptides with Membrane Models (Articolo in rivista) (Prodotto della ricerca)
- Bradykinin antagonists modified with dipeptide mimetic beta-turn inducers (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Impurity analysis of retinoic acid samples (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and enzymatic evaluation of novel partially fluorinated thiol dual ACE/NEP inhibitors (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and molecular modelling studies of prenylated pyrazolines as MAO-B inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Enantioselective synthesis and vanilloid activity evaluation of 1-beta-(p-methoxycinnamoyl)polygodial, an antinociceptive compound from Drymis winteri barks. (Articolo in rivista) (Prodotto della ricerca)
- Enantioselective binding of second generation pyrrolobenzoxazepinones to the catalytic ternary complex of HIV-1 RT wild-type and L100I and K103N drug resistant mutants. (Articolo in rivista) (Prodotto della ricerca)
- Praziquantel derivatives I: Modification of the aromatic ring. (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II \"selective\" inhibitor celecoxib. (Articolo in rivista) (Prodotto della ricerca)
- CARBONIC ANHYDRASE INHIBITORS: X-RAY CRYSTALLOGRAPHIC STUDIES FOR THE BINDING OF 5-AMINO-1,3,4-THIADIZOLE-2-SULFONAMIDE AND 5-(4-AMINO-3-CHLORO-5-FLUOROPHENYLSULFONAMIDO)-1,3,4-THIADIAZOLE-2-SULFONAMIDE TO HUMAN ISOFORM II (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties (Articolo in rivista) (Prodotto della ricerca)
- Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of Thr200 and Gln92 for obtaining tight-binding inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Metabolically labile cannabinoid esters: A 'soft drug' approach for the development of cannabinoid-based therapeutic drugs (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological evaluation of new potential inhibitors of N-acylethanolamine hydrolyzing acid amidase. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- N-Hydroxyurea as zinc binding group in matrix metalloproteinase inhibition: mode of binding in a complex with MMP-8. (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological investigation of S-aryl-S-DABO derivatives as HIV-1 inhibitors. (Articolo in rivista) (Prodotto della ricerca)
- Discovery of novel benzimidazolones as potent non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains. (Articolo in rivista) (Prodotto della ricerca)
- Indolyl-pyrrolone as a new scaffold for Pim1 inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Towards novel S-DABOC inhibitors: Synthesis, biological investigation, and molecular modeling studies. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Discovery of potent nucleotide-mimicking competitive inhibitors of hepatitis C virus NS3 helicase. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and alpha4beta2 nicotinic affinity of unichiral 5-(2-pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and alpha4beta2 nicotinic affinity of 2-pyrrolidinylmethoxyimines and prolinal oxime ethers. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes. (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Development of mitochondrial-targeted derivatives o resveratrol. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- 5-(2-Pyrrolidinyl)oxazolidinones and 2-(2-pyrrolidinyl)benzodioxanes: synthesis of all the stereoisomers and alpha4beta2 nicotinic affinity. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Soluble polyphenols: synthesis and bioavailability of 3,4',5-tri(alpha-D-glucose-3-O-succinyl)resveratrol. (Articolo in rivista) (Prodotto della ricerca)
- Novel imidazole-based combretastatin A-4 analogues: Evaluation of their in vitro antitumor activity and molecular modeling study of their binding to the colchicine site of tubulin (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis of All-trans Isomer of Arachidonic Acid and Its Effect on Rabbit Plateled Aggregation (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of new Praziquantel analogues: Potential candidates for the treatment of schistosomiasis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Design of novel alpha7-subtype-preferring nicotinic acetylcholine receptor agonists: application of docking and MM-PBSA computational approaches, synthetic and pharmacological studies (Articolo in rivista) (Prodotto della ricerca)
- Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Evidences for complex formation between L-dabPNA and aegPNA (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and binding affinity at alpha4beta2 and alpha7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Discovery of the first small molecule inhibitor of human DDX3 specifically designed to target the RNA binding site: towards the next generation HIV-1 inhibitors (Articolo in rivista) (Prodotto della ricerca)
- Enzymatic regio- and diastereoselective hydrolysis of peracetylated glycerol- and erhythritol-beta-glucosides (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Glycosynthase-catalysed syntheses at pH below neutrality. (Articolo in rivista) (Prodotto della ricerca)
- (-)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels (Articolo in rivista) (Prodotto della ricerca)
- New highly hydrosoluble and not self-aggregated perylene derivatives with three and four polar side chains as G-quadruplex telomere targeting agents and telomerase inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Natural and synthetic G-quadruplex interactive berberine derivatives. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds (Articolo in rivista) (Prodotto della ricerca)
- Rational design, synthesis and characterization of potent, drug-like monomeric Smac mimetics as pro-apoptotic anticancer agents (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- New tetrazole-based selective anandamide uptake inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The homovanillyl moiety (Articolo in rivista) (Prodotto della ricerca)
- Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Carbonic anhydrase VII is S-glutathionylated without loss of catalytic activity and affinity for sulfonamide inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators (Articolo in rivista) (Prodotto della ricerca)
- Tetrahydro-beta-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels. . (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candidaalbicans and Candida glabrata (Articolo in rivista) (Prodotto della ricerca)
- 3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Kinetic and anion inhibition studies of a beta-carbonic anhydrase (FbiCA 1) from the C-4 plant Flaveria bidentis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- A novel super-potent neurokinin a receptor antagonist containing dehydroalanine (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Synthetic approaches to DNMT inhibitor SGI-1027 and effects on the U937 leukemia cell line. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Anion inhibition studies of two new beta-carbonic anhydrases from the bacterial pathogen Legionella pneumophila (Articolo in rivista) (Prodotto della ricerca)
- Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum-The eta-carbonic anhydrases (Articolo in rivista) (Prodotto della ricerca)
- Synthesis of sulfonamides with effective inhibitory action against Porphyromonas gingivalis gamma-carbonic anhydrase (Articolo in rivista) (Prodotto della ricerca)
- Effect of acyclic monoterpene alcohols and their derivatives on TRP channels (Articolo in rivista) (Prodotto della ricerca)
- Anion inhibition study of the beta-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Sulfonamide inhibition studies of the delta-carbonic anhydrase from the diatom Thalassiosira weissflogii (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Sulfonamide inhibition studies of the gamma-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
- Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB(1) receptors. (Articolo in rivista) (Prodotto della ricerca)
- SYNTHESIS OF CARBAPENEMS VIA METALLOIMINES-ESTER ENOLATES CONDENSATION - A NEW SYNTHESIS OF (+)-1-BETA-METHYL PS-5 (Articolo in rivista) (Prodotto della ricerca)