http://www.cnr.it/ontology/cnr/individuo/prodotto/ID15790
Antitumor extrolites produced by Penicillium species (Articolo in rivista)
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- Antitumor extrolites produced by Penicillium species (Articolo in rivista) (literal)
- Anno
- 2008-01-01T00:00:00+01:00 (literal)
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- Nicoletti R; Ciavatta M.L.; Buommino E.; Tufano M.A. (literal)
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- 1 Council for Research and Experimentation in Agriculture - Research Unit of Scafati, Via Vitiello 108, 84018 Scafati, Italy
2 Institute of Biomolecular Chemistry, C.N.R., Via Campi Flegrei 36, Pozzuoli, Italy
3 Department of Experimental Medicine, the Second University of Naples, Via De Crecchio 7, 80100 Napoli, Italy (literal)
- Titolo
- Antitumor extrolites produced by Penicillium species (literal)
- Abstract
- Biodiversity is increasingly exploited worldwide for the finding of new pharmaceuticals. In relation to a competitive aptitude developed
in many and diverse environments, microorganisms are able to produce secondary metabolites with cytotoxic and antiproliferative
properties that are valuable in the perspective of antitumor drug discovery. Particularly, fungal species in the genus Penicillium represent a
prolific source of biologically active extrolites that in some cases have already disclosed possible relevance for an application in cancer
chemotherapy. Antiproliferative, pro-apoptotic, anti-angiogenic, anti-metastatic, DNA synthesis and cell cycle inhibitory properties of
these compounds are reviewed in the present paper.
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