ChemMedChem

Label

• ChemMedChem (literal)

Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#rivistaDi

• Synthesis and in vitro evaluation of trifluoroethylamine analogues of enkephalines (Articolo in rivista) (Prodotto della ricerca)
• 3D QSAR Models Built on Structure-Based Alignments of Abl Tyrosine Kinase Inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Design, synthesis, and biological evaluation of 2-aminobenzanilide derivatives as potent and selective HDAC inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Carprofen analogues as sirtuin inhibitors: enzyme and cellular studies. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Synthesis and pharmacological activity of a potent inhibitor of the biosynthesis of the endocannabinoid 2-arachidonoylglycerol. (Articolo in rivista) (Prodotto della ricerca)
• Interaction of Artemisinins with Oxyhemoglobin Hb-Fe-II, Hb-Fe-II, CarboxyHb-Fe-II, Heme-Fe-II, and Carboxyheme Fe-II: Significance for Mode of Action and Implications for Therapy of Cerebral Malaria (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• The Fe2+-Mediated Decomposition, PfATP6 Binding, and Antimalarial Activities of Artemisone and Other Artemisinins: The Unlikelihood of C-Centered Radicals as Bioactive Intermediates (Articolo in rivista) (Prodotto della ricerca)
• Slow-, Tight-Binding HIV-1 Reverse Transcriptase Non-Nucleoside Inhibitors Highly Active against Drug-Resistant Mutants. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Synthesis, biological activity, and ADME properties of novel S-DABOs/N-DABOs as HIV reverse transcriptase inhibitors (Articolo in rivista) (Prodotto della ricerca)
• Peptide Containing Aggregates as Selective Nanocarriers for Therapeutics (Articolo in rivista) (Prodotto della ricerca)
• A partial convergence in action of methylene blue and artemisinins: antagonism with chloroquine, a reversal with verapamil, and an insight into the antimalarial activity of chloroquine. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Structure-Activity Relationship Study of 16a-Thiocamptothecins: an Integrated In Vitro and In Silico Approach (Articolo in rivista) (Prodotto della ricerca)
• Toward the discovery of novel anti-HIV drugs. Second-generation inhibitors of the cellular ATPase DDX3 with improved anti-HIV activity: synthesis, structure-activity relationship analysis, cytotoxicity studies, and target validation. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• The trifluoroethylamine function as peptide bond replacement (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Facile Biocatalytic Access to 9-Fluorenylmethyl Polyglycosides: Evaluation of Antiviral Activity on Immunocompetent Cells (Articolo in rivista) (Prodotto della ricerca)
• A Potent Integrin Antagonist from a Small Library of Cyclic RGD Pentapeptide Mimics Including Benzyl-Substituted Azabicycloalkane Amino Acids (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Atomistic-Level Portrayal of Drug-DNA Interplay: A History of Courtships and Meetings Revealed by Molecular Simulations (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Dopamides, Vanillylamides, Ethanolamides, and Arachidonic Acid Amides of Anti-inflammatory and Analgesic Drug Substances as TRPV1 Ligands. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Facile Oxidation of Leucomethylene Blue and Dihydroflavins by Artemisinins: Relationship with Flavoenzyme Function and Antimalarial Mechanism of Action (Articolo in rivista) (Prodotto della ricerca)
• Substrate-Induced Stable Enzyme-Inhibitor Complex Formation Allows Tight Binding of Novel 2-Aminopyrimidin-4(3H)-ones to Drug-Resistant HIV-1 Reverse Transcriptase Mutants. (Articolo in rivista) (Prodotto della ricerca)
• Identification of Small-Molecule Inhibitors of the XendoU Endoribonucleases Family (Articolo in rivista) (Prodotto della ricerca)
• A combination strategy to inhibit Pim-1: synergism between noncompetitive and ATP-competitive inhibitors. (Articolo in rivista) (Prodotto della ricerca)
• Reactions of Antimalarial Peroxides with Each of Leucomethylene Blue and Dihydroflavins: Flavin Reductase and the Cofactor Model Exemplified (Articolo in rivista) (Prodotto della ricerca)
• Carbonic anhydrase inhibitors: binding of indanesulfonamides to the human isoform II (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Delivery of Suramin as an Antiviral Agent through Liposomal Systems (Articolo in rivista) (Prodotto della ricerca)
• Synthesis of Gd and (68) Ga Complexes in Conjugation with a Conformationally Optimized RGD Sequence as Potential MRI and PET Tumor-Imaging Probes (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Cyclic RGD-Containing Functionalized Azabicycloalkane Peptides as Potent Integrin Antagonists for Tumor Targeting (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• On the Metabolically Active Form of Metaglidasen: Improved Synthesis and Investigation of Its Peculiar Activity on Peroxisome Proliferator-Activated Receptors and Skeletal Muscles. (Articolo in rivista) (Prodotto della ricerca)
• tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• A multidisciplinary approach for the identification of novel HIV-1 non-nucleoside reverse transcriptase inhibitors: S-DABOCs and DAVPs. (Articolo in rivista) (Prodotto della ricerca)
• Design, synthesis, biological evaluation, and molecular modeling studies of TIBO-like cyclic sulfones as non-nucleoside HIV-1 reverse transcriptase inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Conformationally constrained CCK8 analogues obtained from a rationally designed peptide library as ligands for cholecystokinin type B receptor. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Probing the Peptidylglycine alpha-Hydroxylating Monooxygenase Active Site with Novel 4-Phenyl-3-butenoic Acid Based Inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• N2-Benzyloxycarbonylguan-9-yl Acetic Acid Derivatives as HIV-1 Reverse Transcriptase Non-Nucleoside Inhibitors with Decreased Loss of Potency Against Common Drug-Resistance Mutations. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Design and synthesis of thiadiazoles and thiazoles targeting the Bcr-Abl T315I mutant: from docking false positives to ATP-noncompetitive inhibitors. (Articolo in rivista) (Prodotto della ricerca)
• Tuning sensitivity in paramagnetic NMR detection of ligand-DNA interaction (Articolo in rivista) (Prodotto della ricerca)
• Dimerizable redox-sensitive triazine-based cationic lipids for in vitro gene delivery (Articolo in rivista) (Prodotto della ricerca)
• Inhibition of Bcr-Abl Phosphorylation and Induction of Apoptosis by Pyrazolo[3,4-d]pyrimidines in Human Leukemia Cells. (Articolo in rivista) (Prodotto della ricerca)
• Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis, Structure-Activity Relationships, and Docking Studies (Part 2). (Articolo in rivista) (Prodotto della ricerca)
• A High-Affinity Carbohydrate-Containing Inhibitor of Matrix Metalloproteinases (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• N-[2-Methyl-5-(triazol-1-yl)phenyl]pyrimidin-2-amine as a Scaffold for the Synthesis of Inhibitors of Bcr-Abl. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Combining computational and biochemical studies for a rationale on the anti-aromatase activity of natural polyphenols (Articolo in rivista) (Prodotto della ricerca)
• Anticancer therapeutics that target selenoenzymes: synthesis, characterization, in vitro cytotoxicity and thioredoxin reductase inhibition of a series of gold(I) complexes containing hydrophilic phosphine ligands (Articolo in rivista) (Prodotto della ricerca)
• A Combinatorial Approach to 2,4,6-Trisubstituted Triazines with Potent Antimalarial Activity: Combining Conventional Synthesis and Microwave-Assistance (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Design, synthesis, and pharmacological characterization of novel spirocyclic quinuclidinyl-Delta2-isoxazoline derivatives as potent and selective agonists of alpha7 nicotinic acetylcholine receptors. (Articolo in rivista) (Prodotto della ricerca)
• Assessing the bioisosterism of the trifluoromethyl group with a protease probe (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• A DNA Methyltransferase Modulator Inspired by Peyssonenyne Natural Product Structures. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)

Alternative label

• ChemMedChem (literal)
• ChemMedChem. (literal)

Language

• eng (literal)

Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#issn

• 1860-7179 (literal)

Preferred label

• ChemMedChem (literal)

Publisher

• Wiley-VCH-Verl.. Weinheim : DEU (literal)

Incoming links:

Rivista

• Peptide Containing Aggregates as Selective Nanocarriers for Therapeutics (Articolo in rivista) (Prodotto della ricerca)
• Facile Biocatalytic Access to 9-Fluorenylmethyl Polyglycosides: Evaluation of Antiviral Activity on Immunocompetent Cells (Articolo in rivista) (Prodotto della ricerca)
• A High-Affinity Carbohydrate-Containing Inhibitor of Matrix Metalloproteinases (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Combining computational and biochemical studies for a rationale on the anti-aromatase activity of natural polyphenols (Articolo in rivista) (Prodotto della ricerca)
• Assessing the bioisosterism of the trifluoromethyl group with a protease probe (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Synthesis and in vitro evaluation of trifluoroethylamine analogues of enkephalines (Articolo in rivista) (Prodotto della ricerca)
• Dopamides, Vanillylamides, Ethanolamides, and Arachidonic Acid Amides of Anti-inflammatory and Analgesic Drug Substances as TRPV1 Ligands. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• A multidisciplinary approach for the identification of novel HIV-1 non-nucleoside reverse transcriptase inhibitors: S-DABOCs and DAVPs. (Articolo in rivista) (Prodotto della ricerca)
• Substrate-Induced Stable Enzyme-Inhibitor Complex Formation Allows Tight Binding of Novel 2-Aminopyrimidin-4(3H)-ones to Drug-Resistant HIV-1 Reverse Transcriptase Mutants. (Articolo in rivista) (Prodotto della ricerca)
• Design and synthesis of thiadiazoles and thiazoles targeting the Bcr-Abl T315I mutant: from docking false positives to ATP-noncompetitive inhibitors. (Articolo in rivista) (Prodotto della ricerca)
• Inhibition of Bcr-Abl Phosphorylation and Induction of Apoptosis by Pyrazolo[3,4-d]pyrimidines in Human Leukemia Cells. (Articolo in rivista) (Prodotto della ricerca)
• Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: Synthesis, Structure-Activity Relationships, and Docking Studies (Part 2). (Articolo in rivista) (Prodotto della ricerca)
• Identification of Small-Molecule Inhibitors of the XendoU Endoribonucleases Family (Articolo in rivista) (Prodotto della ricerca)
• Conformationally constrained CCK8 analogues obtained from a rationally designed peptide library as ligands for cholecystokinin type B receptor. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Carbonic anhydrase inhibitors: binding of indanesulfonamides to the human isoform II (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Synthesis and pharmacological activity of a potent inhibitor of the biosynthesis of the endocannabinoid 2-arachidonoylglycerol. (Articolo in rivista) (Prodotto della ricerca)
• The trifluoroethylamine function as peptide bond replacement (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• 3D QSAR Models Built on Structure-Based Alignments of Abl Tyrosine Kinase Inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• N2-Benzyloxycarbonylguan-9-yl Acetic Acid Derivatives as HIV-1 Reverse Transcriptase Non-Nucleoside Inhibitors with Decreased Loss of Potency Against Common Drug-Resistance Mutations. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• N-[2-Methyl-5-(triazol-1-yl)phenyl]pyrimidin-2-amine as a Scaffold for the Synthesis of Inhibitors of Bcr-Abl. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Slow-, Tight-Binding HIV-1 Reverse Transcriptase Non-Nucleoside Inhibitors Highly Active against Drug-Resistant Mutants. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Toward the discovery of novel anti-HIV drugs. Second-generation inhibitors of the cellular ATPase DDX3 with improved anti-HIV activity: synthesis, structure-activity relationship analysis, cytotoxicity studies, and target validation. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Anticancer therapeutics that target selenoenzymes: synthesis, characterization, in vitro cytotoxicity and thioredoxin reductase inhibition of a series of gold(I) complexes containing hydrophilic phosphine ligands (Articolo in rivista) (Prodotto della ricerca)
• A Potent Integrin Antagonist from a Small Library of Cyclic RGD Pentapeptide Mimics Including Benzyl-Substituted Azabicycloalkane Amino Acids (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Interaction of Artemisinins with Oxyhemoglobin Hb-Fe-II, Hb-Fe-II, CarboxyHb-Fe-II, Heme-Fe-II, and Carboxyheme Fe-II: Significance for Mode of Action and Implications for Therapy of Cerebral Malaria (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Structure-Activity Relationship Study of 16a-Thiocamptothecins: an Integrated In Vitro and In Silico Approach (Articolo in rivista) (Prodotto della ricerca)
• Cyclic RGD-Containing Functionalized Azabicycloalkane Peptides as Potent Integrin Antagonists for Tumor Targeting (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Facile Oxidation of Leucomethylene Blue and Dihydroflavins by Artemisinins: Relationship with Flavoenzyme Function and Antimalarial Mechanism of Action (Articolo in rivista) (Prodotto della ricerca)
• Reactions of Antimalarial Peroxides with Each of Leucomethylene Blue and Dihydroflavins: Flavin Reductase and the Cofactor Model Exemplified (Articolo in rivista) (Prodotto della ricerca)
• A partial convergence in action of methylene blue and artemisinins: antagonism with chloroquine, a reversal with verapamil, and an insight into the antimalarial activity of chloroquine. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Design, synthesis, and pharmacological characterization of novel spirocyclic quinuclidinyl-Delta2-isoxazoline derivatives as potent and selective agonists of alpha7 nicotinic acetylcholine receptors. (Articolo in rivista) (Prodotto della ricerca)
• The Fe2+-Mediated Decomposition, PfATP6 Binding, and Antimalarial Activities of Artemisone and Other Artemisinins: The Unlikelihood of C-Centered Radicals as Bioactive Intermediates (Articolo in rivista) (Prodotto della ricerca)
• A Combinatorial Approach to 2,4,6-Trisubstituted Triazines with Potent Antimalarial Activity: Combining Conventional Synthesis and Microwave-Assistance (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Dimerizable redox-sensitive triazine-based cationic lipids for in vitro gene delivery (Articolo in rivista) (Prodotto della ricerca)
• Tuning sensitivity in paramagnetic NMR detection of ligand-DNA interaction (Articolo in rivista) (Prodotto della ricerca)
• Design, synthesis, biological evaluation, and molecular modeling studies of TIBO-like cyclic sulfones as non-nucleoside HIV-1 reverse transcriptase inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Synthesis of Gd and (68) Ga Complexes in Conjugation with a Conformationally Optimized RGD Sequence as Potential MRI and PET Tumor-Imaging Probes (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• A DNA Methyltransferase Modulator Inspired by Peyssonenyne Natural Product Structures. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Design, synthesis, and biological evaluation of 2-aminobenzanilide derivatives as potent and selective HDAC inhibitors. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Probing the Peptidylglycine alpha-Hydroxylating Monooxygenase Active Site with Novel 4-Phenyl-3-butenoic Acid Based Inhibitors (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Synthesis, biological activity, and ADME properties of novel S-DABOs/N-DABOs as HIV reverse transcriptase inhibitors (Articolo in rivista) (Prodotto della ricerca)
• tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• A combination strategy to inhibit Pim-1: synergism between noncompetitive and ATP-competitive inhibitors. (Articolo in rivista) (Prodotto della ricerca)
• Carprofen analogues as sirtuin inhibitors: enzyme and cellular studies. (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Delivery of Suramin as an Antiviral Agent through Liposomal Systems (Articolo in rivista) (Prodotto della ricerca)
• Atomistic-Level Portrayal of Drug-DNA Interplay: A History of Courtships and Meetings Revealed by Molecular Simulations (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells (Articolo in rivista) (http://www.cnr.it/ontology/cnr/individuo/prodotto/TIPO1101)
• On the Metabolically Active Form of Metaglidasen: Improved Synthesis and Investigation of Its Peculiar Activity on Peroxisome Proliferator-Activated Receptors and Skeletal Muscles. (Articolo in rivista) (Prodotto della ricerca)