A Nanoparticulate drug delivery system for rivastigmine: physico-chemical and in vitro biological characterization (Articolo in rivista)

Type
Label
  • A Nanoparticulate drug delivery system for rivastigmine: physico-chemical and in vitro biological characterization (Articolo in rivista) (literal)
Anno
  • 2008-01-01T00:00:00+01:00 (literal)
Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#doi
  • 10.1002/mabi.200700165 (literal)
Alternative label
  • E.F. Craparo, G. Pitarresi, M.L. Bondì, M.P. Casaletto, M. Licciardi and G. Giammona (2008)
    A Nanoparticulate drug delivery system for rivastigmine: physico-chemical and in vitro biological characterization
    in Macromolecular bioscience (Print); Wiley-VCH Verlag Gmbh, Weinheim (Germania)
    (literal)
Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#autori
  • E.F. Craparo, G. Pitarresi, M.L. Bondì, M.P. Casaletto, M. Licciardi and G. Giammona (literal)
Pagina inizio
  • 247 (literal)
Pagina fine
  • 259 (literal)
Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#numeroVolume
  • 8 (literal)
Rivista
Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#pagineTotali
  • 13 (literal)
Note
  • ISI Web of Science (WOS) (literal)
Http://www.cnr.it/ontology/cnr/pubblicazioni.owl#affiliazioni
  • Dipartimento di Chimica e Tecnologie Farmaceutiche, Unipa (literal)
Titolo
  • A Nanoparticulate drug delivery system for rivastigmine: physico-chemical and in vitro biological characterization (literal)
Abstract
  • The preparation and characterization of surface-PEGylated polymeric nanoparticles are described. These systems were obtained by UV irradiation of PHM and PHM-PEG2000 as an inverse microemulsion, using an aqueous solution of the PHM/PHM-PEG2000 copolymer mixture as the internal phase and triacetin saturated with water as the external phase, and characterized by dimensional analysis, zeta-potential measurements and XPS. in vitro biological tests demonstrated their cell compatibility and their ability to escape from phagocytosis. Rivastigmine was encapsulated into the nanoparticle structure and drug-release profiles from loaded samples were investigated in PBS at pH¼7.4 and human plasma. (literal)
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